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Intelligence-assisted Structure-Based Drug Discovery\uff0cAISBDD\uff09\u6280\u672f\u81ea\u4e3b\u7814\u53d1\u7684\u80f0\u6dc0\u7d20\u53d7\u4f53\u6fc0\u52a8\u5242\u591a\u80bd\u3002ASC36\u53e3\u670d\u7247\u5242\u7531\u6b4c\u793c\u5229\u7528\u5176\u4e13\u6709\u7684\u53e3\u670d\u591a\u80bd\u9012\u9001\u589e\u5f3a\u6280\u672f\uff08Peptide Oral Transport ENhancement Technology\uff0cPOTENT\uff09\u5f00\u53d1\u5e76\u4f18\u5316\u800c\u6210\uff0c\u8be5\u6280\u672f\u7528\u4e8e\u5b9e\u73b0\u53e3\u670d\u591a\u80bd\u9012\u9001\u3002<\/p>\n<p>\u5728\u975e\u4eba\u7075\u957f\u7c7b\u52a8\u7269\u4e2d\uff0c10\u6beb\u514bASC36\u53e3\u670d\u7247\u5728\u6bcf\u53ea\u52a8\u7269\u4e2d\u6bcf\u65e5\u4e00\u6b21\u7ed9\u836f\uff0c\u7ed9\u836f7\u5929\u540e\uff0c\u7a33\u6001\u4e0b\u7684\u7edd\u5bf9\u53e3\u670d\u751f\u7269\u5229\u7528\u5ea6\uff08absolute oral bioavailability\uff09[1]\u4e3a8%\uff0c\u6d88\u9664\u534a\u8870\u671f\uff08elimination 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advantages in manufacturing\uff09\u3002<\/p>\n<div>\n<p class=\"prnml4\"><span class=\"prnews_span\">[1] 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Technology\uff0cPOTENT\uff09\uff0c\u6b4c\u793c\u5df2\u81ea\u4e3b\u7814\u53d1\u591a\u6b3e\u5c0f\u5206\u5b50\u548c\u591a\u80bd\u5019\u9009\u836f\u7269\uff0c\u5305\u62ec\u5176\u6838\u5fc3\u9879\u76eeASC30\uff0c\u4e00\u6b3e\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u5c0f\u5206\u5b50GLP-1R\u6fc0\u52a8\u5242\uff0c\u7528\u4e8e\u957f\u671f\u4f53\u91cd\u7ba1\u7406\u548c\u7cd6\u5c3f\u75c5\u6cbb\u7597\uff1bASC30_48FDC\uff0c\u4e00\u6b3e\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u5c0f\u5206\u5b50\u53cc\u9776\u70b9\u6fc0\u52a8\u5242\uff0c\u4e3aASC30\uff08GLP-1R\u6fc0\u52a8\u5242\uff09\u4e0eASC48\uff08GIPR\u6fc0\u52a8\u5242\uff09\u7684\u56fa\u5b9a\u5242\u91cf\u590d\u65b9\u5236\u5242\uff1bASC30_48_39FDC\uff0c\u4e00\u6b3e\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u5c0f\u5206\u5b50\u4e09\u9776\u70b9\u6fc0\u52a8\u5242\uff0c\u4e3aASC30\uff08GLP-1R\u6fc0\u52a8\u5242\uff09\u3001ASC48\uff08GIPR\u6fc0\u52a8\u5242\uff09\u4e0eASC39\uff08\u80f0\u6dc0\u7d20\u9009\u62e9\u6027\u53d7\u4f53\u6fc0\u52a8\u5242\uff08SARA\uff09\uff09\u7684\u56fa\u5b9a\u5242\u91cf\u590d\u65b9\u5236\u5242\uff1bASC39\uff0c\u4e00\u6b3e\u4e0eeloralintide\u7c7b\u4f3c\u3001\u5f3a\u6548\u7684\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u5c0f\u5206\u5b50\u80f0\u6dc0\u7d20\u9009\u62e9\u6027\u53d7\u4f53\u6fc0\u52a8\u5242\uff08SARA\uff09\uff1bASC30_39FDC\uff0c\u4e00\u6b3e\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\u5c0f\u5206\u5b50\u53cc\u9776\u70b9\u6fc0\u52a8\u5242\uff0c\u4e3aASC30\uff08GLP-1R\u6fc0\u52a8\u5242\uff09\u4e0eASC39\uff08\u80f0\u6dc0\u7d20\u9009\u62e9\u6027\u53d7\u4f53\u6fc0\u52a8\u5242\uff08SARA\uff09\uff09\u7684\u56fa\u5b9a\u5242\u91cf\u590d\u65b9\u5236\u5242\uff1bASC36\uff0c\u4e00\u6b3e\u80f0\u6dc0\u7d20\u591a\u80bd\uff0c\u8bbe\u8ba1\u4e3a\u6bcf\u6708\u4e00\u6b21\u81f3\u6bcf\u5b63\u5ea6\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u4ee5\u53ca\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\uff1bASC35\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04GLP-1R\/GIPR\u53cc\u9776\u70b9\u6fc0\u52a8\u5242\u591a\u80bd\uff1bASC36_35FDC\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u4e09\u9776\u70b9\u591a\u80bd\u6fc0\u52a8\u5242\uff0c\u4e3aASC36\uff08\u80f0\u6dc0\u7d20\u53d7\u4f53\u6fc0\u52a8\u5242\uff09\u4e0eASC35\uff08GLP-1R\/GIPR\u6fc0\u52a8\u5242\uff09\u7684\u56fa\u5b9a\u5242\u91cf\u590d\u65b9\u5236\u5242\uff1bASC37\uff0c\u4e00\u6b3eGLP-1R\/GIPR\/GCGR\u4e09\u9776\u70b9\u6fc0\u52a8\u5242\u591a\u80bd\uff0c\u8bbe\u8ba1\u4e3a\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u53ca\u6bcf\u65e5\u4e00\u6b21\u53e3\u670d\uff1b\u4ee5\u53caASC36_37FDC\uff0c\u4e00\u6b3e\u6bcf\u6708\u4e00\u6b21\u76ae\u4e0b\u6ce8\u5c04\u56db\u9776\u70b9\u6fc0\u52a8\u5242\u591a\u80bd\uff0c\u4e3aASC36\uff08\u80f0\u6dc0\u7d20\u53d7\u4f53\u6fc0\u52a8\u5242\uff09\u4e0eASC37\uff08GLP-1R\/GIPR\/GCGR\u6fc0\u52a8\u5242\uff09\u7684\u56fa\u5b9a\u5242\u91cf\u590d\u65b9\u5236\u5242\uff0c\u7528\u4e8e\u957f\u671f\u4f53\u91cd\u7ba1\u7406\u3002\u6b4c\u793c\u5df2\u5728\u9999\u6e2f\u8054\u4ea4\u6240\u4e0a\u5e02\uff081672.HK\uff09\u3002<\/p>\n<p>\u6b32\u4e86\u89e3\u66f4\u591a\u4fe1\u606f\uff0c\u656c\u8bf7\u767b\u5f55\u7f51\u7ad9\uff1a<a href=\"http:\/\/www.ascletis.com\/\" target=\"_blank\" rel=\"noopener\">www.ascletis.com<\/a>\u3002<\/p>\n<p>\u8be6\u60c5\u5782\u8be2\uff1a<\/p>\n<p>Peter Vozzo<br \/>ICR Healthcare<br \/>443-231-0505 (\u7f8e\u56fd)<br \/><a href=\"mailto:Peter.vozzo@icrhealthcare.com\" target=\"_blank\" rel=\"noopener\">Peter.vozzo@icrhealthcare.com<\/a>\u00a0<\/p>\n<p>\u6b4c\u793c\u5236\u836f\u6709\u9650\u516c\u53f8PR\u548cIR\u56e2\u961f<br \/>+86-181-0650-9129 (\u4e2d\u56fd)<br \/><a href=\"mailto:pr@ascletis.com\" target=\"_blank\" rel=\"noopener\">pr@ascletis.com<\/a> <br \/><a href=\"mailto:ir@ascletis.com\" target=\"_blank\" rel=\"noopener\">ir@ascletis.com<\/a>\u00a0<\/p>\n<p>\u00a0<\/p>\n<p>SOURCE \u6b4c\u793c\u5236\u836f\u6709\u9650\u516c\u53f8<\/p>","protected":false},"excerpt":{"rendered":"<p>&#8211; \u8be5\u7814\u7a76\u662f\u6b4c\u793c\u4eca\u5e74\u7684\u7b2c\u56db\u9879\u591a\u80bd\u7c7bI\u671f\u7814\u7a76\u3002 &#8211; 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kg\/m\u00b2\uff09\u53d7\u8bd5\u8005\u4e2d\uff0c\u5355\u5242\u91cf\u548c\u591a\u5242\u91cf\u9012\u589e\u53e3\u670d\u7ed9\u836f\u540e\u7684\u5b89\u5168\u6027\u3001\u8010\u53d7\u6027\u3001\u836f\u4ee3\u52a8\u529b\u5b66\u548c\u836f\u6548\u52a8\u529b\u5b66\u3002 &#8220;2026\u5e74\uff0c\u6211\u4eec\u5c31\u591a\u80bd\u7ba1\u7ebf\u542f\u52a8\u4e86\u56db\u9879I\u671f\u7814\u7a76\uff0cASC36\u53e3\u670d\u7247\u662f\u5176\u4e2d\u7b2c\u56db\u9879\u4e5f\u662f\u6700\u65b0\u7684\u4e00\u9879\uff0c\u8fd9\u662f\u6b4c\u793c\u591a\u80bd\u7ba1\u7ebf\u7684\u4e00\u9879\u91cd\u8981\u91cc\u7a0b\u7891\uff0c\u4e5f\u8fdb\u4e00\u6b65\u9a8c\u8bc1\u4e86\u6211\u4eec\u4e13\u6709\u7684POTENT\u53e3\u670d\u591a\u80bd\u9012\u9001\u6280\u672f\u3002&#8221;\u6b4c\u793c\u521b\u59cb\u4eba\u3001\u8463\u4e8b\u4f1a\u4e3b\u5e2d\u517c\u9996\u5e2d\u6267\u884c\u5b98\u5434\u52b2\u6893\u535a\u58eb\u8868\u793a\uff0c&#8221;ASC36\u5728\u4e34\u5e8a\u524d\u7814\u7a76\u4e2d\u8868\u73b0\u51fa\u4ee4\u4eba\u9f13\u821e\u7684\u51cf\u91cd\u7597\u6548\u3001\u826f\u597d\u7684\u53e3\u670d\u751f\u7269\u5229\u7528\u5ea6\u548c\u8f83\u957f\u7684\u534a\u8870\u671f\u3002\u6211\u4eec\u76f8\u4fe1\uff0c\u4e00\u6b3e\u6709\u6548\u7684\u53e3\u670d\u80f0\u6dc0\u7d20\u53d7\u4f53\u6fc0\u52a8\u5242\u6709\u671b\u4e3a\u80a5\u80d6\u4eba\u7fa4\u63d0\u4f9b\u4fbf\u6377\u4e14\u5dee\u5f02\u5316\u7684\u6cbb\u7597\u9009\u62e9\u3002\u7ed3\u5408\u6211\u4eec\u7684\u53e3\u670d\u5c0f\u5206\u5b50\u548c\u957f\u6548\u6ce8\u5c04\u5242\u9879\u76ee\uff0cASC36\u8fdb\u4e00\u6b65\u5f3a\u5316\u4e86\u6211\u4eec\u7684\u591a\u5143\u5316\u4ea7\u54c1\u7ba1\u7ebf\uff0c\u4ee5\u6ee1\u8db3\u80a5\u80d6\u75c7\u53ca\u5176\u4ed6\u4ee3\u8c22\u75be\u75c5\u60a3\u8005\u4e0d\u65ad\u53d8\u5316\u7684\u6cbb\u7597\u9700\u6c42\u3002&#8221; 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